Acetic Acid

Acetic Acid

SCHEMBL6430767

CC(=O)O.CN1CCN(C2CCC(n3nc(-c4ccc(Oc5ccc(CNC(=O)c6ccccc6)cc5)cc4)c4c(N)ncnc43)CC2)CC1

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BTK Q06187 10/20 0.72
LCK P06239 7/20 0.72
SRC P12931 7/20 0.72
TEK Q02763 7/20 0.72
KDR P35968 3/20 0.72
NUDT14 O95848 2/20 0.62
NUDT5 Q9UKK9 2/20 0.62
EGFR P00533 9/20 0.59
LIMK1 P53667 1/20 0.57
LIMK2 P53671 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL6430777 1.00 BTK (0.72) BTKLCKSRCTEKKDR
Acetic Acid SCHEMBL6431629 0.93 LCK (0.74) BTKLCKSRCTEKKDR
Acetic Acid SCHEMBL6431633 0.93 LCK (0.74) BTKLCKSRCTEKKDR
SCHEMBL6431295 0.92 LCK (0.72) BTKLCKSRCTEKKDR
SCHEMBL6431292 0.92 LCK (0.72) BTKLCKSRCTEKKDR
Acetic Acid SCHEMBL6432590 0.92 LCK (0.72) BTKLCKSRCTEKKDR
Acetic Acid SCHEMBL6432593 0.92 LCK (0.72) BTKLCKSRCTEKKDR
SCHEMBL6623451 0.91 LCK (0.77) BTKLCKSRCTEKKDR
SCHEMBL6623453 0.91 LCK (0.77) BTKLCKSRCTEKKDR
Acetic Acid SCHEMBL6430318 0.88 LCK (0.72) BTKLCKSRCTEKKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6921763-B2 Pyrazolopyrimidines as therapeutic agents ABBOTT LABORATORIES (US) 2005-07-26 US disclosed
US-20050008640-A1 Method of treating transplant rejection ABBOTT LABORATORIES 2005-01-13 US disclosed
US-6660744-B1 Kinase inhibitors ABBOTT GMBH & CO. KG (DE) 2003-12-09 US disclosed
EP-1212327-B1 PYRAZOLOPYRIMIDINES AS THERAPEUTIC AGENTS BASF AG (DE) 2003-08-20 EP disclosed
US-20020156081-A1 Pyrazolopyrimidines as therapeutic agents ABBOTT LABORATORIES (US) 2002-10-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050008640-A1 Method of treating transplant rejection LCK, ZAP70, FYN BTK 42/4885LCK 1/4885SRC 46/4885
US-20020156081-A1 Pyrazolopyrimidines as therapeutic agents DPYD, CYP2D6, UGT1A1 BTK 1020/4885LCK 1011/4885SRC 1834/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.