SCHEMBL6430841

SCHEMBL6430841

COCCOc1cc2nccc(Nc3cc(O)c(C)cc3F)c2cc1OC

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 9/20 0.80
FGFR1 P11362 7/20 0.80
KDR P35968 10/20 0.69
RET P07949 4/20 0.59
KIF5B P33176 4/20 0.59
FLT4 P35916 3/20 0.58
FGFR2 P21802 1/20 0.58
FGFR4 P22455 1/20 0.58
FGFR3 P22607 1/20 0.58
EGFR P00533 5/20 0.50
GAK O14976 2/20 0.49
SRC P12931 3/20 0.47
RAF1 P04049 2/20 0.47
BRAF P15056 2/20 0.47
BMPR1B O00238 1/20 0.47
EPHB6 O15197 1/20 0.47
RIPK2 O43353 1/20 0.47
ABL1 P00519 1/20 0.47
LCK P06239 1/20 0.47
EPHA1 P21709 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6431075 0.99 FLT1 (0.79) FLT1FGFR1KDRRETKIF5B
SCHEMBL6434212 0.92 KDR (0.68) FLT1FGFR1KDRRETKIF5B
Hydrochloric Acid SCHEMBL6434300 0.91 KDR (0.67) FLT1FGFR1KDRRETKIF5B
SCHEMBL6432152 0.89 FLT1 (1.00) FLT1FGFR1KDRRETKIF5B
Hydrochloric Acid SCHEMBL6431098 0.88 FLT1 (0.98) FLT1FGFR1KDRRETKIF5B
SCHEMBL6431742 0.87 FLT1 (0.61) FLT1FGFR1KDRRETKIF5B
Hydrochloric Acid SCHEMBL6431020 0.86 FLT1 (0.61) FLT1FGFR1KDRRETKIF5B
SCHEMBL6431128 0.85 EHMT2 (0.64) FLT1FGFR1KDRRETKIF5B
SCHEMBL1194359 0.85 KDR (0.81) FLT1FGFR1KDRRETKIF5B
Hydrochloric Acid SCHEMBL6430760 0.85 EHMT2 (0.63) FLT1FGFR1KDRRETKIF5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP claimed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US claimed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP claimed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO claimed
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed