SCHEMBL6431363

SCHEMBL6431363

COc1cc2nccc(Oc3cc(O)c(C)cc3F)c2cc1OC

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SRC P12931 2/20 0.57
TGFBR1 P36897 2/20 0.57
PDGFRA P16234 5/20 0.53
PDGFRB P09619 1/20 0.53
FGFR2 P21802 1/20 0.53
KDR P35968 5/20 0.52
RET P07949 1/20 0.52
FGFR1 P11362 1/20 0.52
FLT1 P17948 1/20 0.52
KIF5B P33176 1/20 0.52
MET P08581 1/20 0.49
AXL P30530 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6436231 0.90 SRC (0.57) SRCTGFBR1PDGFRAPDGFRBFGFR2
SCHEMBL6431273 0.82 AXL (0.73) SRCPDGFRAPDGFRBFGFR2KDR
SCHEMBL15338419 0.81 SRC (0.70) SRCTGFBR1PDGFRAPDGFRBFGFR2
SCHEMBL24444602 0.81 SRC (0.55) SRCTGFBR1PDGFRAPDGFRBFGFR2
SCHEMBL14742900 0.80 PDGFRA (0.56) SRCTGFBR1PDGFRAPDGFRBFGFR2
SCHEMBL13787639 0.79 SRC (0.61) SRCTGFBR1PDGFRAPDGFRBFGFR2
SCHEMBL6431497 0.79 FLT3 (0.42) SRCTGFBR1KDRRETFGFR1
SCHEMBL6434212 0.78 KDR (0.68) SRCPDGFRAKDRRETFGFR1
SCHEMBL13739661 0.78 SRC (0.60) SRCTGFBR1PDGFRAPDGFRBFGFR2
SCHEMBL20216775 0.78 FGFR2 (0.55) PDGFRAPDGFRBFGFR2KDRAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP claimed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO claimed
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed