SCHEMBL6436231

SCHEMBL6436231

COc1cc2nccc(Oc3cc(O)c(F)cc3C)c2cc1OC

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SRC P12931 2/20 0.57
TGFBR1 P36897 2/20 0.57
PDGFRA P16234 5/20 0.53
PDGFRB P09619 1/20 0.53
KDR P35968 4/20 0.52
FLT1 P17948 1/20 0.50
AURKB Q96GD4 1/20 0.50
FGFR2 P21802 1/20 0.50
MET P08581 1/20 0.49
AXL P30530 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6431363 0.90 SRC (0.57) SRCTGFBR1PDGFRAPDGFRBKDR
SCHEMBL4481865 0.78 SRC (0.60) SRCTGFBR1PDGFRAPDGFRBKDR
SCHEMBL15338419 0.78 SRC (0.70) SRCTGFBR1PDGFRAPDGFRBKDR
SCHEMBL3895983 0.78 SRC (0.69) SRCTGFBR1PDGFRAPDGFRBKDR
SCHEMBL13739661 0.78 SRC (0.60) SRCTGFBR1PDGFRAPDGFRBKDR
SCHEMBL13787639 0.77 SRC (0.61) SRCTGFBR1PDGFRAPDGFRBKDR
Hydrochloric Acid SCHEMBL3893940 0.76 SRC (0.67) SRCTGFBR1PDGFRAPDGFRBKDR
SCHEMBL3894663 0.76 PDGFRB (0.64) SRCTGFBR1PDGFRAPDGFRBFGFR2
SCHEMBL5221950 0.76 EGFR (0.55) SRCTGFBR1PDGFRAPDGFRBKDR
SCHEMBL4400367 0.76 PDGFRB (0.72) SRCTGFBR1PDGFRAPDGFRBFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed