SCHEMBL6431467

SCHEMBL6431467

COc1cc2c(Nc3cc(O[Si](c4ccccc4)(c4ccccc4)C(C)(C)C)c(Cl)cc3F)ccnc2cc1O

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 4/20 0.54
FGFR1 P11362 3/20 0.54
SRC P12931 3/20 0.49
RAF1 P04049 4/20 0.44
BRAF P15056 4/20 0.44
KDR P35968 3/20 0.44
MAPK14 Q16539 1/20 0.42
MET P08581 1/20 0.41
EGFR P00533 6/20 0.41
BRD4 O60885 1/20 0.41
BRD2 P25440 1/20 0.41
BRD3 Q15059 1/20 0.41
GAK O14976 1/20 0.39
FGFR2 P21802 1/20 0.39
FGFR4 P22455 1/20 0.39
FGFR3 P22607 1/20 0.39
FLT4 P35916 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6432661 0.88 FLT1 (0.55) FLT1FGFR1SRCKDRMAPK14
SCHEMBL7452247 0.87 MAPK14 (0.58) FLT1FGFR1SRCRAF1BRAF
SCHEMBL6431182 0.86 EGFR (0.54) FLT1FGFR1SRCKDRMAPK14
SCHEMBL6434966 0.84 FLT1 (0.51) FLT1FGFR1SRCKDRMAPK14
SCHEMBL6432013 0.82 FLT1 (0.49) FLT1FGFR1SRCKDRMAPK14
SCHEMBL8711202 0.82 RAF1 (0.37) FLT1FGFR1SRCRAF1BRAF
SCHEMBL6432009 0.81 SRC (0.45) FLT1FGFR1SRCKDRMAPK14
SCHEMBL6431462 0.81 FLT1 (0.51) FLT1FGFR1SRCRAF1BRAF
SCHEMBL6431016 0.80 EGFR (0.53) FLT1FGFR1SRCBRAFKDR
Hydrochloric Acid SCHEMBL6435465 0.78 FLT1 (0.83) FLT1FGFR1SRCRAF1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed