SCHEMBL6432009

SCHEMBL6432009

COc1cc2c(Nc3cc(O[Si](c4ccccc4)(c4ccccc4)C(C)(C)C)c(Cl)cc3F)ccnc2cc1OC(C)c1ncc[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 4/20 0.45
FGFR1 P11362 2/20 0.45
FLT1 P17948 2/20 0.45
KDR P35968 1/20 0.41
EGFR P00533 6/20 0.39
MET P08581 1/20 0.38
GAK O14976 2/20 0.37
MAPK14 Q16539 1/20 0.37
KRAS P01116 2/20 0.36
SOS1 Q07889 2/20 0.36
AXL P30530 4/20 0.35
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35
BMPR1B O00238 1/20 0.35
EPHB6 O15197 1/20 0.35
RIPK2 O43353 1/20 0.35
ABL1 P00519 1/20 0.35
LCK P06239 1/20 0.35
EPHA1 P21709 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8509887 0.84 SRC (0.43) SRCFGFR1FLT1KDREGFR
Hydrochloric Acid SCHEMBL6434139 0.84 FLT1 (0.63) SRCFGFR1FLT1KDREGFR
SCHEMBL6432661 0.83 FLT1 (0.55) SRCFGFR1FLT1KDREGFR
SCHEMBL6432187 0.83 FLT1 (0.64) SRCFGFR1FLT1KDREGFR
SCHEMBL6431182 0.82 EGFR (0.54) SRCFGFR1FLT1KDREGFR
SCHEMBL6431467 0.81 FLT1 (0.54) SRCFGFR1FLT1KDREGFR
SCHEMBL6434966 0.80 FLT1 (0.51) SRCFGFR1FLT1KDREGFR
SCHEMBL6432013 0.77 FLT1 (0.49) SRCFGFR1FLT1KDREGFR
SCHEMBL6431016 0.76 EGFR (0.53) SRCFGFR1FLT1KDREGFR
SCHEMBL7451653 0.71 EGFR (0.59) SRCFGFR1FLT1KDREGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed