SCHEMBL6432008

SCHEMBL6432008

COc1cc2c(Nc3cc(O[SiH2]C(C)(C)C(c4ccccc4)c4ccccc4)c(Cl)cc3F)ccnc2cc1OCc1nccn1C

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 6/20 0.46
FGFR1 P11362 5/20 0.46
EGFR P00533 4/20 0.45
SRC P12931 3/20 0.43
KDR P35968 9/20 0.42
RET P07949 1/20 0.42
EPHA2 P29317 4/20 0.40
ERBB2 P04626 3/20 0.40
EPHB4 P54760 2/20 0.40
MAPK14 Q16539 1/20 0.37
MET P08581 1/20 0.36
FGFR2 P21802 2/20 0.35
FGFR4 P22455 2/20 0.35
FGFR3 P22607 2/20 0.35
FLT4 P35916 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7460007 0.91 RET (0.52) FLT1FGFR1EGFRKDRRET
SCHEMBL6431180 0.89 EGFR (0.55) FLT1FGFR1EGFRSRCKDR
SCHEMBL6432660 0.88 FLT1 (0.51) FLT1FGFR1EGFRSRCKDR
SCHEMBL6434962 0.87 EGFR (0.51) FLT1FGFR1EGFRSRCKDR
SCHEMBL6432013 0.84 FLT1 (0.49) FLT1FGFR1EGFRSRCKDR
SCHEMBL6431462 0.83 FLT1 (0.51) FLT1FGFR1EGFRSRCKDR
SCHEMBL6431014 0.83 EGFR (0.50) FLT1FGFR1EGFRSRCKDR
SCHEMBL6432182 0.80 FLT1 (0.70) FLT1FGFR1EGFRSRCKDR
SCHEMBL8509887 0.80 SRC (0.43) FLT1FGFR1EGFRSRCKDR
SCHEMBL7451650 0.79 EGFR (0.54) FLT1FGFR1EGFRSRCKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed