SCHEMBL6434962

SCHEMBL6434962

COc1cc2c(Nc3cc(O[SiH2]C(C)(C)C(c4ccccc4)c4ccccc4)c(Cl)cc3F)ccnc2cc1OCc1ccncc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.51
FLT1 P17948 8/20 0.48
FGFR1 P11362 4/20 0.48
KDR P35968 10/20 0.48
SRC P12931 3/20 0.45
EPHA2 P29317 4/20 0.44
ERBB2 P04626 2/20 0.44
GAK O14976 1/20 0.39
EPHB4 P54760 2/20 0.39
MAPK14 Q16539 1/20 0.38
FLT4 P35916 2/20 0.36
FGFR2 P21802 1/20 0.36
FGFR4 P22455 1/20 0.36
FGFR3 P22607 1/20 0.36
MET P08581 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6431180 0.96 EGFR (0.55) EGFRFLT1FGFR1KDRSRC
SCHEMBL6432660 0.90 FLT1 (0.51) EGFRFLT1FGFR1KDRSRC
SCHEMBL6432008 0.87 FLT1 (0.46) EGFRFLT1FGFR1KDRSRC
SCHEMBL7451650 0.86 EGFR (0.54) EGFRFLT1FGFR1KDRSRC
SCHEMBL6431462 0.86 FLT1 (0.51) EGFRFLT1FGFR1KDRSRC
SCHEMBL6431014 0.83 EGFR (0.50) EGFRFLT1FGFR1KDRSRC
SCHEMBL6434966 0.83 FLT1 (0.51) EGFRFLT1FGFR1KDRSRC
SCHEMBL8509887 0.82 SRC (0.43) EGFRFLT1FGFR1KDRSRC
SCHEMBL7450324 0.81 KDR (0.63) EGFRFLT1FGFR1KDRSRC
SCHEMBL6433880 0.79 FLT1 (0.75) EGFRFLT1FGFR1KDRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed