SCHEMBL6433044

SCHEMBL6433044

CCOC(=O)C[C@H](NCCN(CCCc1ccc2c(n1)NCCC2)C(=O)OC(C)(C)C)c1ccc(OC)nc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.55
ITGB3 P05106 19/20 0.55
ITGB6 P18564 7/20 0.49
ITGB1 P05556 2/20 0.48
ITGA5 P08648 2/20 0.48
ITGA2B P08514 3/20 0.47
ITGB8 P26012 3/20 0.47
ITGB5 P18084 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6433042 1.00 ITGAV (0.55) ITGAVITGB3ITGB6ITGB1ITGA5
SCHEMBL6304539 0.95 ITGAV (0.57) ITGAVITGB3ITGB6ITGB1ITGA5
SCHEMBL6304533 0.95 ITGAV (0.57) ITGAVITGB3ITGB6ITGB1ITGA5
SCHEMBL6435940 0.85 ITGAV (0.53) ITGAVITGB3ITGB6ITGB1ITGA2B
SCHEMBL6435942 0.85 ITGAV (0.53) ITGAVITGB3ITGB6ITGB1ITGA2B
SCHEMBL6303755 0.85 ITGAV (0.60) ITGAVITGB3ITGB6ITGB1ITGA5
SCHEMBL6303762 0.85 ITGAV (0.60) ITGAVITGB3ITGB6ITGB1ITGA5
SCHEMBL6222793 0.80 ITGAV (0.49) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL6433481 0.79 ITGAV (0.49) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL7587385 0.79 ITGAV (0.40) ITGAVITGB3ITGB6ITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040111-B1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2005-06-22 EP disclosed
US-6017926-A Integrin receptor antagonists MERCK & CO., INC. (US) 2000-01-25 US disclosed