SCHEMBL6433481

SCHEMBL6433481

CCOC(=O)CN(CCCc1ccc2c(n1)NCCC2)C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.49
ITGB6 P18564 10/20 0.49
ITGB3 P05106 14/20 0.44
ITGA2B P08514 4/20 0.44
ITGB5 P18084 4/20 0.44
ITGB8 P26012 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6222793 0.92 ITGAV (0.49) ITGAVITGB6ITGB3ITGA2BITGB5
SCHEMBL6431911 0.85 ITGAV (0.52) ITGAVITGB6ITGB3ITGA2BITGB5
SCHEMBL19465186 0.84 ITGAV (0.57) ITGAVITGB6ITGB3ITGA2BITGB5
SCHEMBL6225569 0.84 ITGAV (0.51) ITGAVITGB6ITGB3ITGA2BITGB5
SCHEMBL6222791 0.83 ITGAV (0.51) ITGAVITGB6ITGB3ITGA2BITGB5
SCHEMBL6265738 0.80 ITGAV (0.56) ITGAVITGB6ITGB3ITGA2BITGB5
SCHEMBL6433042 0.79 ITGAV (0.55) ITGAVITGB6ITGB3ITGA2BITGB5
SCHEMBL6433044 0.79 ITGAV (0.55) ITGAVITGB6ITGB3ITGA2BITGB5
SCHEMBL19809630 0.79 ITGAV (0.61) ITGAVITGB6ITGB3ITGA2BITGB5
SCHEMBL6435940 0.78 ITGAV (0.53) ITGAVITGB6ITGB3ITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040111-B1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2005-06-22 EP disclosed
US-6017926-A Integrin receptor antagonists MERCK & CO., INC. (US) 2000-01-25 US disclosed