SCHEMBL6434256

SCHEMBL6434256

COc1cc2c(Nc3ccc(Cl)cc3F)ccnc2cc1OCCO

nearest known ligand 0.83

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 14/20 0.83
KDR P35968 13/20 0.83
FGFR1 P11362 12/20 0.83
SRC P12931 3/20 0.64
FLT4 P35916 6/20 0.61
EGFR P00533 6/20 0.61
EPHB2 P29323 1/20 0.58
FGFR2 P21802 1/20 0.55
FGFR4 P22455 1/20 0.55
FGFR3 P22607 1/20 0.55
NUDT1 P36639 2/20 0.53
CSF1R P07333 1/20 0.53
ERBB2 P04626 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6431606 0.95 FLT1 (0.81) FLT1KDRFGFR1SRCFLT4
SCHEMBL6431198 0.91 FLT1 (1.00) FLT1KDRFGFR1SRCFLT4
Hydrochloric Acid SCHEMBL6431524 0.90 FLT1 (0.98) FLT1KDRFGFR1SRCFLT4
Hydrochloric Acid SCHEMBL6434964 0.89 FLT1 (0.82) FLT1KDRFGFR1SRCFLT4
Hydrochloric Acid SCHEMBL6436544 0.87 FLT1 (0.79) FLT1KDRFGFR1SRCFLT4
SCHEMBL6430988 0.87 FLT1 (0.79) FLT1KDRFGFR1SRCFLT4
SCHEMBL7867708 0.85 FLT1 (0.83) FLT1KDRFGFR1FLT4EGFR
SCHEMBL27530372 0.84 KDR (0.66) FLT1KDRFGFR1SRCFLT4
Trifluoroacetic Acid SCHEMBL1889530 0.84 FLT1 (0.71) FLT1KDRFGFR1SRCFLT4
SCHEMBL6998899 0.84 FLT1 (0.74) FLT1KDRFGFR1SRCFLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP claimed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US claimed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP claimed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO claimed
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed