SCHEMBL6435408

SCHEMBL6435408

O=C(O)C[C@@H](c1cccnc1)N1CCN(CCCc2ccc3c(n2)NCCC3)C1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 1.00
ITGB3 P05106 18/20 1.00
ITGB6 P18564 4/20 0.75
ITGA2B P08514 4/20 0.75
ITGB8 P26012 3/20 0.75
ITGB1 P05556 1/20 0.75
ITGA5 P08648 1/20 0.75
ITGB5 P18084 4/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6432332 1.00 ITGAV (1.00) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL6432340 1.00 ITGAV (1.00) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL6432128 0.89 ITGAV (0.80) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL6431937 0.89 ITGAV (0.80) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL6431734 0.89 ITGAV (0.80) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL6432134 0.88 ITGAV (0.82) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL6433437 0.88 ITGAV (0.82) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL6432131 0.88 ITGAV (0.82) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL6431872 0.88 ITGAV (0.80) ITGAVITGB3ITGB6ITGA2BITGB8
SCHEMBL25665881 0.88 ITGAV (0.80) ITGAVITGB3ITGB6ITGA2BITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040111-B1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2005-06-22 EP claimed
EP-1040111-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-10-04 EP claimed
WO-1999031099-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO claimed
EP-1040111-B1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2005-06-22 EP disclosed
EP-1040111-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-10-04 EP disclosed
US-6017926-A Integrin receptor antagonists MERCK & CO., INC. (US) 2000-01-25 US disclosed
WO-1999031099-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed