SCHEMBL6435484

SCHEMBL6435484

COCCOc1cc2nccc(Oc3cc(OCc4ccccc4)c(C)cc3F)c2cc1C#N

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MET P08581 14/20 0.41
KDR P35968 2/20 0.41
MST1R Q04912 2/20 0.41
FLT3 P36888 1/20 0.38
AXL P30530 2/20 0.38
HGF P14210 1/20 0.38
RET P07949 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6431497 0.84 FLT3 (0.42) METKDRFLT3AXLRET
SCHEMBL2178142 0.80 XDH (0.41) KDR
SCHEMBL6098451 0.76 KDR (0.47) METKDRMST1RRET
SCHEMBL1891898 0.76 XDH (0.41) KDR
SCHEMBL14540955 0.76 FNTA (0.46) METFLT3AXL
SCHEMBL1892973 0.75 MAOB (0.42) METKDRAXL
SCHEMBL1893599 0.75 MAOB (0.42) METKDRAXL
SCHEMBL14540937 0.75 SRC (0.44) KDR
SCHEMBL1895977 0.74 AXL (0.45) METKDRFLT3AXL
SCHEMBL6431297 0.74 AXL (0.67) METKDRMST1RFLT3AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929526-B1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ASTRAZENECA AB (SE) 2005-07-27 EP disclosed
US-6809097-B1 ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY ZENECA LIMITED (GB) 2004-10-26 US disclosed
EP-0929526-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1999-07-21 EP disclosed
WO-1998013350-A1 QINOLINE DERIVATIVES INHIBITING THE EFFECT OF GROWTH FACTORS SUCH AS VEGF ZENECA LIMITED (GB) 1998-04-02 WO disclosed