SCHEMBL6435751

SCHEMBL6435751

O=Cc1cc(Br)c(F)cc1I

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 7/20 0.39
PRKDC P78527 1/20 0.34
PTPN1 P18031 1/20 0.32
LMNA P02545 1/20 0.32
CYP2A6 P11509 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31466810 0.94 ERN1 (0.41) ERN1PRKDCPTPN1LMNACYP2A6
SCHEMBL30952047 0.83 ERN1 (0.35) ERN1PRKDCLMNA
SCHEMBL29655114 0.80 ERN1 (0.43) ERN1PRKDCPTPN1LMNA
SCHEMBL933374 0.80 ERN1 (0.43) ERN1PRKDCPTPN1LMNA
SCHEMBL633623 0.78 ERN1 (0.45) ERN1PRKDCPTPN1LMNA
SCHEMBL28880933 0.77 PRKDC (0.44) ERN1PRKDCLMNA
SCHEMBL24485242 0.75 TDP1 (0.42) ERN1PRKDCPTPN1LMNA
SCHEMBL874654 0.75 ERN1 (0.48) ERN1
SCHEMBL29712897 0.75 TDP1 (0.42) ERN1PRKDCPTPN1LMNA
SCHEMBL31477129 0.75 GRIA1 (0.41) ERN1PRKDCPTPN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194429-B1 POTASSIUM CHANNEL OPENERS ABBOTT LAB (US) 2005-03-30 EP disclosed
US-6593335-B1 Disease than can be ameliorated with a potassium channel opener in a host mammal, comprising administering to the mammal in need thereof a therapeutically effective amount of the compound of claim 1; said disease is epilepsy, Raynaud's ABBOTT LABORATORIES 2003-07-15 US disclosed
EP-1194429-A1 POTASSIUM CHANNEL OPENERS Abbott Laboratories (US) 2002-04-10 EP disclosed
WO-2000078768-A1 POTASSIUM CHANNEL OPENERS ABBOTT LABORATORIES (US) 2000-12-28 WO disclosed