SCHEMBL6437376

SCHEMBL6437376

COc1nc(Oc2cccc(F)c2)c(-c2ccc(Cl)cc2)c(-c2cc(Cl)cc(Cl)c2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.45
CNR2 P34972 5/20 0.45
MAT2A P31153 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HTT P42858 1/20 0.39
F10 P00742 1/20 0.35
NR1H2 P55055 1/20 0.35
ALDH1A1 P00352 3/20 0.34
HPGD P15428 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
USP2 O75604 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
MRGPRX1 Q96LB2 1/20 0.33
CYP2C9 P11712 1/20 0.33
MAPK1 P28482 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4803482 0.87 CNR1 (0.58) CNR1CNR2MAT2A
SCHEMBL6440656 0.80 GAA (0.36) CNR1CNR2MAT2AHTTALDH1A1
SCHEMBL4810139 0.79 CNR1 (0.56) CNR1CNR2MEN1KMT2AHTT
SCHEMBL4808039 0.77 CNR1 (0.56) CNR1CNR2
SCHEMBL4804629 0.75 CNR1 (0.56) CNR1CNR2MEN1KMT2AALDH1A1
SCHEMBL4807322 0.74 CNR1 (0.57) CNR1CNR2
SCHEMBL4802298 0.72 CNR1 (0.54) CNR1CNR2
SCHEMBL4807346 0.70 CNR1 (0.44) CNR1CNR2MAT2ACYP1A2CYP3A4
SCHEMBL6439861 0.70 CNR1 (0.45) CNR1CNR2MEN1KMT2AALDH1A1
SCHEMBL4807031 0.68 CNR1 (0.53) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546115-A2 SUBSTITUTED PYRIMIDINES Merck & Co., Inc. (US) 2005-06-29 EP disclosed
WO-2004029204-A2 SUBSTITUTED PYRIMIDINES MERCK & CO., INC. (US) 2004-04-08 WO disclosed