SCHEMBL6440656

SCHEMBL6440656

COc1nc(Oc2cncc(Cl)c2)c(-c2ccc(Cl)cc2)c(-c2cc(Cl)cc(Cl)c2)n1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
MAT2A P31153 1/20 0.36
CNR1 P21554 2/20 0.34
CNR2 P34972 2/20 0.34
PPARG P37231 1/20 0.34
SCN2A Q99250 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4801891 0.87 CNR1 (0.45) MAT2ACNR1CNR2PPARG
SCHEMBL6437376 0.80 CNR1 (0.45) GAAHTTMAT2ACNR1CNR2
SCHEMBL4808021 0.78 CNR1 (0.43) CNR1CNR2PPARG
SCHEMBL4807346 0.74 CNR1 (0.44) MAT2ACNR1CNR2NPSR1
SCHEMBL4804629 0.70 CNR1 (0.56) CNR1CNR2ALDH1A1MAPTHPGD
SCHEMBL4808039 0.70 CNR1 (0.56) CNR1CNR2
SCHEMBL4807100 0.69 CNR1 (0.47) CNR1CNR2
SCHEMBL4807322 0.69 CNR1 (0.57) CNR1CNR2
SCHEMBL6454643 0.68 CNR1 (0.33) CNR1CNR2
SCHEMBL4807155 0.68 CNR1 (0.46) MAT2ACNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546115-A2 SUBSTITUTED PYRIMIDINES Merck & Co., Inc. (US) 2005-06-29 EP disclosed
WO-2004029204-A2 SUBSTITUTED PYRIMIDINES MERCK & CO., INC. (US) 2004-04-08 WO disclosed