SCHEMBL6440478

SCHEMBL6440478

O=C(c1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CCC(N2C[CH]CCC2)C(c2ccc(F)cc2)C1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 11/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ATM Q13315 1/20 0.42
HSD11B1 P28845 2/20 0.42
RHOA P61586 5/20 0.41
RHOC P08134 3/20 0.41
TACR2 P21452 3/20 0.41
TACR3 P29371 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6440125 0.90 NPC1 (0.46) TACR1NPC1RAB9AATMHSD11B1
SCHEMBL6440129 0.90 NPC1 (0.46) TACR1NPC1RAB9AATMHSD11B1
SCHEMBL5918177 0.86 TACR1 (0.43) TACR1NPC1RAB9AATMHSD11B1
SCHEMBL6441184 0.86 RHOA (0.45) TACR1NPC1RAB9AATMHSD11B1
SCHEMBL6439779 0.86 TACR1 (0.43) TACR1NPC1RAB9AATMHSD11B1
SCHEMBL5918155 0.83 HSD11B1 (0.44) TACR1NPC1RAB9AATMHSD11B1
SCHEMBL6439954 0.83 SLC18A3 (0.44) TACR1NPC1RAB9AATMHSD11B1
SCHEMBL5802584 0.83 TACR1 (0.47) TACR1HSD11B1RHOARHOCTACR2
SCHEMBL5918148 0.83 TACR1 (0.47) TACR1HSD11B1RHOARHOCTACR2
SCHEMBL6439955 0.83 SLC18A3 (0.44) TACR1NPC1RAB9AATMHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1360184-B1 PIPERIDINE DERIVATIVES AS NEUROKININ 1 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2005-03-30 EP disclosed