SCHEMBL6441759

SCHEMBL6441759

CCOC(=O)c1cc(Br)c(F)c(Cl)c1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.46
CYP4A11 Q02928 1/20 0.46
MAOB P27338 1/20 0.45
TSHR P16473 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
KDM4E B2RXH2 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
BAZ2B Q9UIF8 1/20 0.42
BAZ2A Q9UIF9 1/20 0.42
CA1 P00915 4/20 0.42
CA2 P00918 4/20 0.42
CA12 O43570 3/20 0.42
CA9 Q16790 3/20 0.42
CA7 P43166 2/20 0.41
CA14 Q9ULX7 2/20 0.41
GPR35 Q9HC97 1/20 0.40
MAPK1 P28482 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9328789 0.84 CYP4F2 (0.48) CYP4F2CYP4A11TSHRNPSR1KDM4E
SCHEMBL4501337 0.84 TSHR (0.46) CYP4F2CYP4A11TSHRNPSR1KDM4E
SCHEMBL4468897 0.82 KMT2A (0.40) CYP4F2CYP4A11MAOBNPSR1KDM4E
SCHEMBL6439456 0.80 TSHR (0.42) CYP4F2CYP4A11TSHRNPSR1KDM4E
SCHEMBL6841276 0.78 CYP4F2 (0.52) CYP4F2CYP4A11MAOBTSHRNPSR1
SCHEMBL71222 0.77 TSHR (0.57) CYP4F2CYP4A11MAOBTSHRNPSR1
SCHEMBL4627413 0.77 TSHR (0.57) CYP4F2CYP4A11MAOBTSHRNPSR1
SCHEMBL4625497 0.77 CYP4F2 (0.54) CYP4F2CYP4A11MAOBTSHRNPSR1
SCHEMBL1819905 0.77 TSHR (0.48) CYP4F2CYP4A11MAOBTSHRNPSR1
SCHEMBL4465988 0.76 ALDH1A1 (0.38) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045823-B1 PROCESS FOR MAKING CERTAIN BENZOIC ACID COMPOUNDS PROCTER & GAMBLE (US) 2005-11-02 EP disclosed
US-6348624-B1 TREATING 1-BROMO-2,4-DIFLUOROBENZENE WITH STRONG, NON-NUCLEOPHILIC BASE, REACTING WITH ELECTROPHILIC REAGENT, TREATING WITH ALKALI OR ALKALINE EARTH METAL OR ORGANOMETALLIC REAGENT AND CARBON DIOXIDE, OR FORMYLATING AND OXIDIZING THE PROCTER & GAMBLE CO. 2002-02-19 US disclosed
CN-1284939-A Process for making certain benzoic acid compounds PROCTER & GAMBLE (US) 2001-02-21 CN disclosed
EP-1045823-A1 PROCESS FOR MAKING CERTAIN BENZOIC ACID COMPOUNDS THE PROCTER & GAMBLE COMPANY (US) 2000-10-25 EP disclosed
WO-1999035117-A1 PROCESS FOR MAKING CERTAIN BENZOIC ACID COMPOUNDS THE PROCTER & GAMBLE COMPANY (US) 1999-07-15 WO disclosed