SCHEMBL6441892

SCHEMBL6441892

O=C(NCCc1c[nH]c2ccccc12)Oc1ccc(F)c2c(C(=O)C(=O)N3CCN(C(=O)c4ccccc4)CC3)c[nH]c12

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.51
HTR1B P28222 2/20 0.51
HTR2A P28223 2/20 0.51
HTR2C P28335 2/20 0.51
HTR2B P41595 2/20 0.51
FAAH O00519 2/20 0.48
LMNA P02545 1/20 0.45
CYP2C9 P11712 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
PTGS2 P35354 1/20 0.42
CYP3A4 P08684 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
KDM4E B2RXH2 1/20 0.41
SIRT1 Q96EB6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6445354 0.87 CYP2C9 (0.50) HTR1AHTR1BHTR2AHTR2CHTR2B
SCHEMBL6442987 0.85 CYP2C9 (0.49) HTR1AHTR1BHTR2AHTR2CHTR2B
SCHEMBL6458040 0.85 CYP2C9 (0.49) HTR1AHTR1BHTR2AHTR2CHTR2B
SCHEMBL6442418 0.84 CYP2C9 (0.51) LMNACYP2C9CYP3A4MAPTKDM4E
SCHEMBL6443286 0.84 CYP2C9 (0.49) HTR1AHTR1BHTR2AHTR2CHTR2B
SCHEMBL6442104 0.82 CYP2C9 (0.53) CYP2C9RAB9ACYP3A4KDM4E
SCHEMBL6445721 0.82 CYP2C9 (0.45) LMNACYP2C9CYP3A4
SCHEMBL6440978 0.81 CYP2C9 (0.54) CYP2C9RAB9ACYP3A4KDM4E
SCHEMBL6444101 0.81 CYP2C9 (0.56) LMNACYP2C9RAB9ACYP3A4MAPT
SCHEMBL6442978 0.81 CYP2C9 (0.51) LMNACYP2C9MEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299382-B1 COMPOSITION AND ANTIVIRAL ACTIVITY OF SUBSTITUTED INDOLEOXOACETIC PIPERAZINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2005-09-21 EP claimed