SCHEMBL6442978

SCHEMBL6442978

COC(CNC(=O)Oc1ccc(F)c2c(C(=O)C(=O)N3CCN(C(=O)c4ccccc4)CC3)c[nH]c12)OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.51
CYP3A4 P08684 4/20 0.46
CYP2C19 P33261 6/20 0.45
CYP2D6 P10635 5/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C8 P10632 1/20 0.45
CYP2B6 P20813 1/20 0.45
KCNH2 Q12809 1/20 0.45
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
ACHE P22303 1/20 0.33
BACE1 P56817 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
DPP4 P27487 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALOX15 P16050 1/20 0.33
BTK Q06187 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6442418 0.88 CYP2C9 (0.51) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL6445354 0.88 CYP2C9 (0.50) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL6444101 0.87 CYP2C9 (0.56) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL6442104 0.87 CYP2C9 (0.53) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL6442987 0.87 CYP2C9 (0.49) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL6440978 0.86 CYP2C9 (0.54) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL6443286 0.85 CYP2C9 (0.49) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL6442045 0.83 CYP2C9 (0.56) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL6446934 0.83 ALDH1A1 (0.49) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2
SCHEMBL6441328 0.83 CYP2C9 (0.46) CYP2C9CYP3A4CYP2C19CYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299382-B1 COMPOSITION AND ANTIVIRAL ACTIVITY OF SUBSTITUTED INDOLEOXOACETIC PIPERAZINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2005-09-21 EP claimed