SCHEMBL6441933

SCHEMBL6441933

C[C@H](Oc1nc(N)nc(-c2cc(Br)co2)c1C#N)c1ccccn1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 18/20 0.38
ADORA2A P29274 17/20 0.38
ADORA2B P29275 4/20 0.38
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
FFAR2 O15552 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6440919 0.84 ADORA2A (0.56) ADORA1ADORA2AADORA2BKDM4EMEN1
SCHEMBL7145343 0.82 ADORA1 (0.41) ADORA1ADORA2AADORA2BKDM4EMEN1
SCHEMBL5040238 0.76 SQOR (0.37) ADORA1ADORA2AADORA2BALDH1A1POLB
SCHEMBL6444873 0.70 ADORA1 (0.34) ADORA1ADORA2AADORA2BKDM4EALDH1A1
SCHEMBL5139767 0.70 ADORA1 (0.43) ADORA1ADORA2AADORA2BKDM4EMEN1
SCHEMBL5133351 0.69 TLR7 (0.38) ADORA1ADORA2AADORA2BKDM4EMEN1
SCHEMBL6442327 0.69 HSP90AA1 (0.33) ALDH1A1POLB
SCHEMBL6443293 0.68 CYP1A2 (0.49) ADORA1ADORA2AADORA2BKDM4EMEN1
SCHEMBL6444534 0.68 ADORA2A (0.55) ADORA1ADORA2AADORA2BKDM4EMEN1
Pyridine SCHEMBL7881098 0.68 ADORA1 (0.40) ADORA1ADORA2AADORA2BKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1261327-B1 ADENOSINE RECEPTOR MODULATORS HOFFMANN LA ROCHE (CH) 2005-04-27 EP disclosed