SCHEMBL6444147

SCHEMBL6444147

CC(C)C(c1c(C(=O)O)ccc(C(=O)O)c1C(C(C)C)C(C)C)C(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
ALDH1A1 P00352 6/20 0.44
ALOX15 P16050 1/20 0.40
MAPT P10636 3/20 0.38
HDAC8 Q9BY41 2/20 0.38
SELL P14151 1/20 0.38
SELP P16109 1/20 0.38
ACE2 Q9BYF1 1/20 0.38
TSHR P16473 2/20 0.37
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA7 P43166 2/20 0.37
CA9 Q16790 2/20 0.37
CA14 Q9ULX7 2/20 0.37
HAAO P46952 1/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28798325 0.86 ALDH1A1 (0.48) ALDH1A1ALOX15MAPTHDAC8TSHR
SCHEMBL6444165 0.82 ACE2 (0.38) CYP1A2ALDH1A1ALOX15MAPTHDAC8
SCHEMBL1950385 0.80 CYP1A2 (0.50) CYP1A2ALDH1A1ALOX15MAPTHDAC8
SCHEMBL728753 0.78 CYP1A2 (0.48) CYP1A2ALDH1A1ALOX15MAPTHDAC8
SCHEMBL17797891 0.73 ALDH1A1 (0.46) CYP1A2ALDH1A1ALOX15MAPTHDAC8
SCHEMBL28238364 0.73 CYP1A2 (0.42) CYP1A2ALDH1A1ALOX15MAPTHDAC8
SCHEMBL6448117 0.73 CYP1A2 (0.42) CYP1A2ALDH1A1ALOX15MAPTACE2
SCHEMBL15123952 0.73 CYP1A2 (0.42) CYP1A2ALDH1A1ALOX15SELLSELP
SCHEMBL3389839 0.71 ALDH1A1 (0.52) ALDH1A1ALOX15MAPTHDAC8TSHR
SCHEMBL6838116 0.71 SELL (0.48) CYP1A2ALDH1A1ALOX15MAPTSELL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194396-B1 SELECTED CYCLOHEXANE-1,3- AND 1,4-DICARBOXYLIC ACID ESTERS BASF AG (DE) 2005-11-09 EP claimed
EP-1194396-B1 SELECTED CYCLOHEXANE-1,3- AND 1,4-DICARBOXYLIC ACID ESTERS BASF AG (DE) 2005-11-09 EP disclosed