SCHEMBL6444947

SCHEMBL6444947

C=CC(CCc1ccccc1)O[Si](C)(C)C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 2/20 0.36
PRSS1 P07477 2/20 0.33
CTSG P08311 2/20 0.33
CTRB1 P17538 2/20 0.33
CMA1 P23946 2/20 0.33
CYP24A1 Q07973 1/20 0.33
BLM P54132 1/20 0.32
TSHR P16473 1/20 0.32
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15184990 1.00 MMP13 (0.36) MMP13PRSS1CTSGCTRB1CMA1
SCHEMBL16414800 0.85 BLM (0.38) PRSS1CTSGCTRB1CMA1CYP24A1
SCHEMBL15271471 0.85 BLM (0.38) PRSS1CTSGCTRB1CMA1CYP24A1
SCHEMBL6449609 0.85 BLM (0.38) PRSS1CTSGCTRB1CMA1CYP24A1
SCHEMBL12549853 0.84 PRSS1 (0.33) PRSS1CTSGCTRB1CMA1CYP24A1
SCHEMBL27318265 0.83 TSHR (0.36) TSHRPPARA
SCHEMBL7552716 0.83 PRSS1 (0.34) PRSS1CTSGCTRB1CMA1CYP24A1
SCHEMBL7552725 0.83 PRSS1 (0.34) PRSS1CTSGCTRB1CMA1CYP24A1
SCHEMBL4494128 0.83 PRSS1 (0.34) PRSS1CTSGCTRB1CMA1CYP24A1
SCHEMBL4494121 0.83 PRSS1 (0.34) PRSS1CTSGCTRB1CMA1CYP24A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0402646-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 1998-07-22 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed