SCHEMBL6447254

SCHEMBL6447254

NCC#Cc1ccccc1C#CCN

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 12/20 0.61
CYP2C9 P11712 10/20 0.61
CYP1A2 P05177 10/20 0.61
CYP3A4 P08684 8/20 0.61
THPO P40225 1/20 0.61
BLM P54132 1/20 0.58
PMP22 Q01453 1/20 0.58
CYP2A6 P11509 12/20 0.47
CYP2E1 P05181 10/20 0.47
CYP2D6 P10635 9/20 0.47
CYP2B6 P20813 9/20 0.47
CYP2C8 P10632 6/20 0.47
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
AOC1 P19801 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2929973 0.85 CYP2C19 (0.56) CYP2C19CYP2C9CYP1A2CYP3A4THPO
SCHEMBL23122854 0.84 CYP2C19 (0.50) CYP2C19CYP2C9CYP1A2CYP3A4THPO
SCHEMBL29745157 0.84 CYP2C19 (0.50) CYP2C19CYP2C9CYP1A2CYP3A4THPO
SCHEMBL8144729 0.84 CYP2C19 (0.55) CYP2C19CYP2C9CYP1A2CYP3A4THPO
SCHEMBL5175910 0.84 CYP2C19 (0.50) CYP2C19CYP2C9CYP1A2CYP3A4THPO
SCHEMBL8144728 0.84 CYP2C19 (0.50) CYP2C19CYP2C9CYP1A2CYP3A4THPO
SCHEMBL7573003 0.80 MEN1 (0.48) CYP2C19CYP2C9CYP1A2CYP3A4THPO
Hydrochloric Acid SCHEMBL21803707 0.79 BLM (0.48) CYP2C19CYP2C9CYP1A2CYP3A4THPO
SCHEMBL29745077 0.79 CYP1A2 (0.58) CYP2C19CYP2C9CYP1A2CYP3A4THPO
SCHEMBL23124208 0.79 CYP1A2 (0.58) CYP2C19CYP2C9CYP1A2CYP3A4THPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6960588-B1 Tryptase inhibitors ALTANA PHARMA AG (DE) 2005-11-01 US disclosed
EP-1216236-A1 TRYPTASE INHIBITORS Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 2002-06-26 EP disclosed
WO-2001019809-A1 TRYPTASE INHIBITORS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2001-03-22 WO disclosed