SCHEMBL6447487

SCHEMBL6447487

N=C(NCCCN)c1cc[c]cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 9/20 0.34
F2 P00734 3/20 0.34
PRSS2 P07478 3/20 0.34
PRSS3 P35030 3/20 0.34
ST14 Q9Y5Y6 3/20 0.34
F10 P00742 1/20 0.34
TMPRSS6 Q8IU80 2/20 0.33
IDO1 P14902 1/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA3 P07451 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CA5B Q9Y2D0 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450887 0.82 SMN1; SMN2 (0.41)
SCHEMBL28278881 0.81 F2 (0.40) F2F10IDO1CA12CA1
SCHEMBL3035405 0.79 CYP1A2 (0.50) GRIN1GRIN2AGRIN2B
SCHEMBL17826868 0.79 PRSS1 (0.37) PRSS1F2PRSS2PRSS3ST14
SCHEMBL15149748 0.79 L3MBTL1 (0.42) PRSS1F2PRSS2PRSS3ST14
SCHEMBL7992188 0.78 L3MBTL1 (0.34) KDM4E
SCHEMBL21168095 0.75 NPC1 (0.51) PRSS1F2PRSS2PRSS3ST14
SCHEMBL18719673 0.75 HPGD (0.46) PRSS1F2PRSS2PRSS3ST14
SCHEMBL549147 0.73 NQO2 (0.50) PRSS1F2PRSS2PRSS3ST14
SCHEMBL7985505 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1545544-A2 COMBINATIONS OF DRUGS FOR THE TREATMENT OF NEOPLASMS Combinatorx, Incorporated (US) 2005-06-29 EP disclosed
WO-2004006842-A2 COMBINATIONS OF DRUGS FOR THE TREATMENT OF NEOPLASMS COMBINATORX, INCORPORATED (US) 2004-01-22 WO disclosed
WO-2004002430-A2 COMBINATIONS FOR THE TREATMENT OF FUNGAL INFECTIONS COMBINATORX INCORPORATED (US) 2004-01-08 WO disclosed