SCHEMBL6447680

SCHEMBL6447680

CC(C)[C@H](NC(=O)OCc1ccccn1)C(=O)N[C@@H](Cc1ccccc1)[C@H](O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)OCc1ccccn1)C(C)C

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.69
CTSD P07339 5/20 0.60
SMN1; SMN2 Q16637 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
MAPT P10636 1/20 0.49
TSHR P16473 1/20 0.49
CASP3 P42574 1/20 0.47
CASP7 P55210 1/20 0.47
NPC1 O15118 1/20 0.47
LMNA P02545 1/20 0.47
RAB9A P51151 1/20 0.47
PGR P06401 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
PTGS1 P23219 1/20 0.47
SLC6A2 P23975 1/20 0.47
REN P00797 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6445023 1.00 CA2 (0.69) CA2CTSDSMN1; SMN2CYP1A2CYP2D6
SCHEMBL7343161 1.00 CA2 (0.69) CA2CTSDSMN1; SMN2CYP1A2CYP2D6
SCHEMBL6449063 1.00 CA2 (0.69) CA2CTSDSMN1; SMN2CYP1A2CYP2D6
SCHEMBL9227910 1.00 CA2 (0.69) CA2CTSDSMN1; SMN2CYP1A2CYP2D6
SCHEMBL7275899 0.98 CA2 (0.66) CA2CTSDSMN1; SMN2CYP1A2CYP2D6
SCHEMBL7270130 0.96 CA2 (0.64) CA2CTSDSMN1; SMN2CYP1A2CYP2D6
SCHEMBL7428656 0.94 CA2 (0.62) CA2CTSDSMN1; SMN2CYP1A2CYP2D6
SCHEMBL7334911 0.94 CA2 (0.62) CA2CTSDSMN1; SMN2CYP1A2CYP2D6
SCHEMBL7330979 0.93 CA2 (0.61) CA2CTSDSMN1; SMN2CYP1A2CYP2D6
SCHEMBL6449444 0.93 CA2 (0.61) CA2CTSDREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP claimed
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0402646-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 1998-07-22 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed