SCHEMBL6448124

SCHEMBL6448124

CC(C)(C)OC(=O)N[C@H](Cc1cccc2ccc(O[Si](c3ccccc3)(c3ccccc3)C(C)(C)C)cc12)C(N)=O

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.52
CTSK P43235 4/20 0.52
PTPN1 P18031 2/20 0.45
CTSB P07858 1/20 0.43
SCN9A Q15858 3/20 0.43
REN P00797 2/20 0.42
NQO2 P16083 1/20 0.41
CCKBR P32239 2/20 0.40
ACE P12821 2/20 0.40
EGLN2 Q96KS0 1/20 0.39
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6455893 0.81 NQO2 (0.61) CTSSCTSKPTPN1CTSBSCN9A
SCHEMBL6469664 0.78 TRPV1 (0.46) CTSSCTSKCTSBNQO2
SCHEMBL7627072 0.78 CTSS (0.42) CTSSCTSKPTPN1CTSB
SCHEMBL7627063 0.78 CTSS (0.42) CTSSCTSKPTPN1CTSB
SCHEMBL8662603 0.76 CTSS (0.62) CTSSCTSKPTPN1CTSBSCN9A
SCHEMBL31385404 0.75 PPARA (0.46) CTSSCTSKCTSBRENACE
SCHEMBL4122289 0.75 CTSS (0.76) CTSSCTSKPTPN1SCN9AACE
SCHEMBL4600435 0.75 CTSS (0.76) CTSSCTSKPTPN1SCN9AACE
SCHEMBL29401990 0.75 CTSS (0.76) CTSSCTSKPTPN1SCN9AACE
SCHEMBL613640 0.75 CTSS (0.76) CTSSCTSKPTPN1SCN9AACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090011-A4 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 2005-04-06 EP disclosed
EP-1090011-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2001-04-11 EP disclosed
WO-2000001701-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2000-01-13 WO disclosed