SCHEMBL6450166

SCHEMBL6450166

CCOC(C(=O)NCc1ccc(C(=N)N)cc1OCC(=O)NCCN(CC)CC)c1c(F)cc(OC)cc1F

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
F10 P00742 5/20 0.59
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP3A4 P08684 1/20 0.42
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HTT P42858 2/20 0.34
TMEM97 Q5BJF2 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
F2 P00734 4/20 0.33
PRSS1 P07477 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TMPRSS15 P98073 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6450173 1.00 F10 (0.59) F10CYP1A2CYP2D6CYP3A4MEN1
Hydrochloric Acid SCHEMBL5037357 0.99 F10 (0.60) F10CYP1A2CYP2D6CYP3A4MEN1
Hydrochloric Acid SCHEMBL5037369 0.99 F10 (0.60) F10CYP1A2CYP2D6CYP3A4MEN1
SCHEMBL5044244 0.90 F10 (0.61) F10F2PRSS1NPSR1TMPRSS15
SCHEMBL5044248 0.90 F10 (0.61) F10F2PRSS1NPSR1TMPRSS15
Hydrochloric Acid SCHEMBL5041040 0.90 F10 (0.63) F10F2PRSS1NPSR1TMPRSS15
Hydrochloric Acid SCHEMBL5041029 0.90 F10 (0.63) F10F2PRSS1NPSR1TMPRSS15
SCHEMBL5045716 0.88 F10 (0.74) F10F2PRSS1
SCHEMBL5045699 0.88 F10 (0.74) F10F2PRSS1
Hydrochloric Acid SCHEMBL5041928 0.87 F10 (0.68) F10F2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567498-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-08-31 EP disclosed
WO-2004048335-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-06-10 WO disclosed