SCHEMBL6455679

SCHEMBL6455679

CN1C(=O)CN=C(c2cccc(C#N)c2)c2cc(-c3ccccc3)ccc21.COc1ccccc1-c1ccc2c(c1)C(c1cccc(C#N)c1)=NCC(=O)N2C

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 8/20 0.64
GABRA5 P31644 8/20 0.64
GABRA2 P47869 8/20 0.64
GABRA3 P34903 7/20 0.64
GABRG2 P18507 6/20 0.64
GABRB3 P28472 6/20 0.64
PDE2A O00408 2/20 0.52
GABRB2 P47870 6/20 0.52
GABRP O00591 1/20 0.49
GABRD O14764 1/20 0.49
CACNA1F O60840 1/20 0.49
ALB P02768 1/20 0.49
GABRB1 P18505 1/20 0.49
OPRK1 P41145 1/20 0.49
AKR1C3 P42330 1/20 0.49
GABRA4 P48169 1/20 0.49
AKR1C2 P52895 1/20 0.49
GABRE P78334 1/20 0.49
CACNA1D Q01668 1/20 0.49
AKR1C1 Q04828 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5034654 0.97 GABRA1 (0.65) GABRA1GABRA5GABRA2GABRA3GABRG2
SCHEMBL5042562 0.91 GABRA1 (0.78) GABRA1GABRA5GABRA2GABRA3GABRG2
SCHEMBL5044341 0.89 GABRA1 (0.64) GABRA1GABRA5GABRA2GABRA3GABRG2
SCHEMBL5034629 0.89 GABRA1 (0.63) GABRA1GABRA5GABRA2GABRA3GABRG2
SCHEMBL5034691 0.89 GABRA1 (0.63) GABRA1GABRA5GABRA2GABRA3GABRG2
SCHEMBL6031148 0.89 PDE2A (0.62) GABRA1GABRA5GABRA2GABRA3GABRG2
SCHEMBL5038976 0.88 GABRA1 (0.64) GABRA1GABRA5GABRA2GABRA3GABRG2
SCHEMBL6031566 0.88 GABRA1 (0.54) GABRA1GABRA5GABRA2GABRA3GABRG2
SCHEMBL5037427 0.88 PDE2A (0.63) GABRA1GABRA5GABRA2GABRA3GABRG2
SCHEMBL5034707 0.88 GABRA1 (0.59) GABRA1GABRA5GABRA2GABRA3GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1548011-A1 Benzo[1,4]diazepin-2-one derivatives as phosphodiesterase PDE2 inhibitors, preparation and therapeutic use thereof NEURO3D (FR) 2005-06-29 EP disclosed