SCHEMBL645773

SCHEMBL645773

CN(Cc1ccon1)S(=O)(=O)c1cc(-c2nnc(O)n2-c2ccccc2Cl)c(O)cc1O

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 4/20 0.48
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
TP53 P04637 1/20 0.31
EIF4E P06730 1/20 0.31
MKNK1 Q9BUB5 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30
MEN1 O00255 1/20 0.30
PKM P14618 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL644537 0.91 HSP90AA1 (0.42) HSP90AA1NPC1POLBPKM
SCHEMBL644652 0.90 HSP90AA1 (0.51) HSP90AA1NPC1RAB9AEIF4EMKNK1
SCHEMBL644517 0.86 HSP90AA1 (0.49) HSP90AA1ALDH1A1LMNAPKM
SCHEMBL646642 0.86 HSP90AA1 (0.52) HSP90AA1TP53ALDH1A1LMNAPOLB
SCHEMBL646966 0.86 HSP90AA1 (0.52) HSP90AA1TP53ALDH1A1LMNAPOLB
SCHEMBL648090 0.85 HSP90AA1 (0.49) HSP90AA1TP53ALDH1A1
SCHEMBL644655 0.85 HSP90AA1 (0.51) HSP90AA1TP53ALDH1A1POLBTSHR
SCHEMBL646290 0.84 HSP90AA1 (0.48) HSP90AA1TP53ALDH1A1LMNAPOLB
SCHEMBL4933407 0.84 HSP90AA1 (0.55) HSP90AA1ALDH1A1LMNATSHRHTT
SCHEMBL646667 0.84 HSP90AA1 (0.51) HSP90AA1TP53ALDH1A1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2023922-B1 TRIAZOLE DERIVATIVES II MERCK PATENT GMBH (DE) 2012-07-11 EP claimed
US-8119795-B2 Triazole derivatives II MERCK PATENT GMBH (DE) 2012-02-21 US claimed
US-20100022540-A1 TRIAZOLE DERIVATIVES II MERCK PATENT GESELLSCHAFT (DE) 2010-01-28 US claimed
EP-2023922-B1 TRIAZOLE DERIVATIVES II MERCK PATENT GMBH (DE) 2012-07-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100022540-A1 TRIAZOLE DERIVATIVES II HSP90AB1, HSP90AA1, HSP90AB2P HSP90AA1 2/4885NPC1 634/4885RAB9A 2229/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.