SCHEMBL6462918

SCHEMBL6462918

CN1CCN(c2ccc(F)cc2/C=C2\CCCN(c3ccc(F)c(F)c3)C2=O)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HDAC3 O15379 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
ADRA1B P35368 1/20 0.37
HDAC1 Q13547 3/20 0.37
LMNA P02545 2/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
IDO2 Q6ZQW0 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
RAB9A P51151 1/20 0.36
BPTF Q12830 1/20 0.35
TSHR P16473 1/20 0.35
POLB P06746 1/20 0.35
MCL1 Q07820 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6430654 1.00 ALDH1A1 (0.42) ALDH1A1L3MBTL1HDAC3HDAC8ADRA1B
SCHEMBL6431119 0.90 ALDH1A1 (0.42) ALDH1A1L3MBTL1HDAC1SMN1; SMN2POLB
SCHEMBL6431123 0.90 ALDH1A1 (0.42) ALDH1A1L3MBTL1HDAC1SMN1; SMN2POLB
SCHEMBL6430942 0.88 MAPT (0.42) ALDH1A1L3MBTL1HDAC1LMNASMN1; SMN2
SCHEMBL6430946 0.88 MAPT (0.42) ALDH1A1L3MBTL1HDAC1LMNASMN1; SMN2
SCHEMBL6430630 0.82 KMT2A (0.43) ALDH1A1L3MBTL1LMNAMEN1KMT2A
SCHEMBL6430629 0.82 KMT2A (0.43) ALDH1A1L3MBTL1LMNAMEN1KMT2A
SCHEMBL6436217 0.82 MAPT (0.43) ALDH1A1L3MBTL1LMNAIDO1TDO2
SCHEMBL6436235 0.82 MAPT (0.43) ALDH1A1L3MBTL1LMNAIDO1TDO2
SCHEMBL6431125 0.77 HDAC1 (0.45) ALDH1A1L3MBTL1ADRA1BHDAC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6924289-B2 Benzyl(Idene)-lactam derivatives, their preparation and their use as selective (ANT) agonists of 5-HT1A- and/or 5-HT1D receptors PFIZER INC (US) 2005-08-02 US claimed
US-6462048-B2 3-(2-(4-METHYLPIPERAZIN-1-YL)-BENZYLIDENE)-1,3-DIHYDRO-INDOL-2-ONE FOR EXAMPLE; USEFUL AS PSYCHOTHERAPEUTIC AGENTS PFIZER INC. 2002-10-08 US disclosed