SCHEMBL6464580

SCHEMBL6464580

COC(=O)c1c(Br)c(C)n(Cc2ccc(C#N)cc2)c1C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.65
CYP11B1 P15538 1/20 0.49
CYP11B2 P19099 1/20 0.49
LMNA P02545 3/20 0.45
KDM4E B2RXH2 2/20 0.45
HTT P42858 2/20 0.45
MAPT P10636 3/20 0.44
TDP1 Q9NUW8 1/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
TSHR P16473 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
KLKB1 P03952 1/20 0.43
KLK1 P06870 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90B1 P14625 1/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 2/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6465312 0.84 AR (0.89) ARCYP11B1CYP11B2LMNAKDM4E
SCHEMBL6469739 0.83 AR (0.52) ARLMNAKDM4EHTTMAPT
SCHEMBL6466362 0.83 AR (0.69) ARLMNAKDM4EHTTMAPT
SCHEMBL6465292 0.80 AR (0.82) ARCYP11B1CYP11B2LMNAKDM4E
SCHEMBL6466721 0.79 AR (0.80) ARCYP11B1CYP11B2LMNAKDM4E
SCHEMBL6468792 0.79 AR (0.80) ARCYP11B1CYP11B2KDM4EMAPT
SCHEMBL6468911 0.79 AR (1.00) ARLMNAMAPTTDP1TSHR
SCHEMBL6469732 0.78 AR (0.82) ARCYP11B1CYP11B2LMNAKDM4E
SCHEMBL6882430 0.78 AR (0.75) ARCYP11B1CYP11B2LMNAKDM4E
SCHEMBL6469313 0.78 AR (0.77) ARCYP11B1CYP11B2LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050101657-A1 Pyrrole derivatives for preventing or treating cancer sensitive to hormones; administered with luteininzing hormone releasing hormone derivative TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 2005-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050101657-A1 Pyrrole derivatives for preventing or treating cancer sensitive to hormones; administered with luteininzing hormone releasing hormone derivative SHBG, PRLHR, FSHR AR 6/4885CYP11B1 145/4885CYP11B2 151/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.