SCHEMBL6464971

SCHEMBL6464971

CCCC(CCNC(=O)O)NC(=O)O

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 16/20 0.42
TAS1R1 Q7RTX1 16/20 0.42
CHRM1 P11229 1/20 0.37
AKR1A1 P14550 1/20 0.37
CHRM3 P20309 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
ADRA1A P35348 1/20 0.37
HRH1 P35367 1/20 0.37
DRD3 P35462 1/20 0.37
SLC6A3 Q01959 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
DPP7 Q9UHL4 1/20 0.34
PLA2G2C Q5R387 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5133204 0.87 TAS1R3 (0.50) TAS1R3TAS1R1CHRM1AKR1A1CHRM3
SCHEMBL17141303 0.87 DPP7 (0.42) TAS1R3TAS1R1DPP7PLA2G2C
SCHEMBL28960765 0.86 CYP2D6 (0.37) TAS1R3TAS1R1ADRA1ATDP1CYP2D6
SCHEMBL28355266 0.85 PLA2G2C (0.47) DPP7PLA2G2C
SCHEMBL6120544 0.79 TAS1R3 (0.44) TAS1R3TAS1R1CHRM1AKR1A1CHRM3
SCHEMBL18063334 0.79 CYP2D6 (0.33) CYP2D6CYP2C19
SCHEMBL20914941 0.79 PLA2G2C (0.51) TAS1R3TAS1R1CHRM1AKR1A1CHRM3
SCHEMBL17112231 0.79 CYP2D6 (0.33) CYP2D6CYP2C19
SCHEMBL6717845 0.79 TAS1R3 (0.50) TAS1R3TAS1R1CHRM1AKR1A1CHRM3
SCHEMBL28681574 0.78 PLA2G10 (0.50) TAS1R3TAS1R1CHRM1AKR1A1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1515702-A1 ABUSE-PROTECTED ADMINISTRATION FORM Grünenthal GmbH (DE) 2005-03-23 EP disclosed
WO-2003105808-A1 ABUSE-PROTECTED ADMINISTRATION FORM Grünenthal GmbH (DE) 2003-12-24 WO disclosed