SCHEMBL6465112

SCHEMBL6465112

CCCC[C@H](NC(=O)CCS(=O)(=O)Cc1ccccc1)C(=O)c1nc2ccccc2o1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 12/20 0.47
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
CTSK P43235 1/20 0.47
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
FAAH O00519 3/20 0.44
CES1 P23141 2/20 0.44
DAGLA Q9Y4D2 1/20 0.44
ALDH1A1 P00352 1/20 0.43
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7187229 0.87 CTSS (0.43) CTSSCTSLCTSBCTSKCYP3A4
SCHEMBL6063897 0.87 KMT2A (0.45) CTSSCTSLCTSBCTSKCYP3A4
SCHEMBL6468436 0.80 CTSS (0.44) CTSSCYP3A4CYP2C9ALDH1A1
SCHEMBL5413826 0.80 CTSS (0.46) CTSSCYP3A4CYP2C9
SCHEMBL6462867 0.78 CTSS (0.41) CTSSCYP3A4CYP2C9ALDH1A1
SCHEMBL6463186 0.77 CTSS (0.50) CTSSCTSLCTSBCTSKCYP3A4
SCHEMBL6466909 0.77 DAGLA (0.56) CTSSCTSLCTSBCTSKCYP3A4
SCHEMBL6466589 0.77 DAGLA (0.56) CTSSCTSLCTSBCTSKCYP3A4
SCHEMBL6464424 0.77 CTSS (0.43) CTSSCYP3A4CYP2C9ALDH1A1
SCHEMBL7049521 0.77 CTSS (0.46) CTSSCTSLCTSBCTSKCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed