SCHEMBL646609

SCHEMBL646609

CC(C)C(c1oc2cc(F)ccc2c(=O)c1Cc1ccccc1)N(CCCN)C(=O)c1onc2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 10/20 0.60
KCNH2 Q12809 2/20 0.60
MAP1LC3B Q9GZQ8 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C19 P33261 1/20 0.37
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
KIF23 Q02241 1/20 0.32
HTT P42858 1/20 0.31
ACP1 P24666 2/20 0.31
PTPN1 P18031 1/20 0.31
KDM4E B2RXH2 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
HSD17B3 P37058 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
ERAP1 Q9NZ08 1/20 0.31
ESR1 P03372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL645676 1.00 KIF11 (0.60) KIF11KCNH2MAP1LC3BCYP3A4CYP2C19
SCHEMBL646890 0.91 KIF11 (0.73) KIF11KCNH2MAP1LC3BCYP3A4CYP2C19
SCHEMBL644968 0.87 KIF11 (0.64) KIF11KCNH2MAP1LC3BCYP3A4CYP2C19
SCHEMBL645263 0.87 KIF11 (0.64) KIF11KCNH2MAP1LC3BCYP3A4CYP2C19
SCHEMBL2456301 0.85 KIF11 (0.62) KIF11KCNH2MAP1LC3BCYP3A4CYP2C19
SCHEMBL644051 0.85 KIF11 (0.70) KIF11KCNH2MAP1LC3BCYP3A4CYP2C19
SCHEMBL646152 0.85 KIF11 (0.65) KIF11KCNH2MAP1LC3BCYP3A4CYP2C19
SCHEMBL646430 0.84 KIF11 (0.83) KIF11KCNH2MAP1LC3BCYP3A4CYP2C19
SCHEMBL644014 0.84 KIF11 (0.73) KIF11KCNH2MAP1LC3BCYP3A4CYP2C19
SCHEMBL645375 0.83 KIF11 (0.65) KIF11KCNH2MAP1LC3BCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119678-B2 Compounds, compositions and methods CYTOKINETICS, INCORPORATED (US) 2012-02-21 US disclosed