SCHEMBL6467155

SCHEMBL6467155

C=S(=C)(C)N(C)c1cc(-c2nnc(C(C)(Cc3ccccc3)NC(=O)OC(C)(C)C)o2)cc(C(=O)OC)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.39
BACE2 Q9Y5Z0 1/20 0.36
NPSR1 Q6W5P4 6/20 0.32
LMNA P02545 5/20 0.32
TSHR P16473 5/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
GAA P10253 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA7 P43166 1/20 0.32
CA14 Q9ULX7 1/20 0.32
CTSS P25774 3/20 0.32
CTSK P43235 2/20 0.32
MAPT P10636 4/20 0.31
ATM Q13315 1/20 0.31
ALDH1A1 P00352 5/20 0.31
HPGD P15428 4/20 0.31
HSD17B10 Q99714 4/20 0.31
HTT P42858 3/20 0.31
PKM P14618 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6468486 0.94 BACE1 (0.40) BACE1BACE2NPSR1LMNATSHR
SCHEMBL2725259 0.93 BACE1 (0.45) BACE1BACE2NPSR1LMNATSHR
SCHEMBL2725260 0.93 BACE1 (0.45) BACE1BACE2NPSR1LMNATSHR
SCHEMBL2727491 0.87 BACE1 (0.46) BACE1BACE2NPSR1LMNATSHR
SCHEMBL2727492 0.87 BACE1 (0.46) BACE1BACE2NPSR1LMNATSHR
SCHEMBL2729373 0.84 NPSR1 (0.35) BACE1NPSR1LMNATSHRSMN1; SMN2
SCHEMBL6467777 0.84 NPSR1 (0.35) BACE1NPSR1LMNATSHRSMN1; SMN2
SCHEMBL2729369 0.84 NPSR1 (0.35) BACE1NPSR1LMNATSHRSMN1; SMN2
SCHEMBL12578538 0.83 BACE1 (0.46) BACE1BACE2NPSR1LMNATSHR
SCHEMBL3588745 0.80 BACE1 (0.58) BACE1BACE2NPSR1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed