SCHEMBL6469671

SCHEMBL6469671

Clc1ncc(CC2CCCNC2)s1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.49
HRH4 Q9H3N8 5/20 0.49
EED O75530 4/20 0.41
ALDH1A1 P00352 1/20 0.39
KCNH2 Q12809 1/20 0.37
USP7 Q93009 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
CCNT1 O60563 1/20 0.35
CHEK1 O14757 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29281499 0.81 HRH3 (0.44) HRH3HRH4ALDH1A1LMNAGAA
SCHEMBL3158557 0.71 HRH3 (0.58) HRH3HRH4EEDKCNH2CHRNB2
SCHEMBL3161259 0.69 HRH3 (0.51) HRH3HRH4EEDKCNH2
SCHEMBL21359085 0.69 HRH3 (0.51) HRH3HRH4EED
SCHEMBL21359086 0.69 HRH3 (0.51) HRH3HRH4EED
SCHEMBL5188074 0.69 EED (0.45) HRH3HRH4EEDKCNH2CCNT1
SCHEMBL20281485 0.69 HRH3 (0.48) HRH3HRH4EEDKCNH2CHEK1
SCHEMBL13576643 0.68 KCNH2 (0.53) HRH3HRH4EEDALDH1A1KCNH2
SCHEMBL13576618 0.68 KCNH2 (0.53) HRH3HRH4EEDALDH1A1KCNH2
Hydrochloric Acid SCHEMBL21358856 0.68 HRH3 (0.50) HRH3HRH4EED

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1495002-A1 BENZAMIDE DERIVATIVES USEFUL AS HISTONE DEACETYLASE INHIBITORS Astrazeneca AB (SE) 2005-01-12 EP disclosed
WO-2003087057-A1 BENZAMIDE DERIVATIVES USEFUL AS HISTONE DEACETYLASE INHIBITORS ASTRAZENECA AB (SE) 2003-10-23 WO disclosed