SCHEMBL6469858

SCHEMBL6469858

CCCc1[nH]c(SC)nc1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.38
HCAR2 Q8TDS4 5/20 0.37
KDM4E B2RXH2 1/20 0.36
KDM6B O15054 1/20 0.36
KDM4A O75164 1/20 0.36
KDM4D Q6B0I6 1/20 0.36
HIF1AN Q9NWT6 1/20 0.36
KDM2A Q9Y2K7 1/20 0.36
CYP2C19 P33261 2/20 0.35
HSD17B10 Q99714 2/20 0.35
ALDH1A1 P00352 2/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CYP2C9 P11712 1/20 0.33
PIN1 Q13526 2/20 0.33
HAO1 Q9UJM8 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GPR84 Q9NQS5 1/20 0.32
USP2 O75604 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6469854 0.86 HCAR2 (0.44) HTTHCAR2KDM4EKDM6BKDM4A
SCHEMBL13646746 0.79 HCAR2 (0.41) HCAR2KDM4ECYP2C19HSD17B10ALDH1A1
SCHEMBL5870591 0.77 HCAR2 (0.38) HCAR2KDM4ECYP2C19HSD17B10PIN1
Formamide SCHEMBL5870611 0.77 HCAR2 (0.39) HCAR2CYP2C19HSD17B10PIN1
SCHEMBL9879081 0.72 HTT (0.49) HTTKDM4ECYP2C19ALDH1A1MAPT
SCHEMBL5870589 0.69 CYP2C19 (0.65) HCAR2KDM4ECYP2C19HSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL5869997 0.68 CYP2C19 (0.62) HCAR2KDM4ECYP2C19HSD17B10ALDH1A1
SCHEMBL15335687 0.67 KDM6B (0.44) HTTKDM4EKDM6BKDM4AKDM4D
SCHEMBL28211381 0.67 HCAR2 (0.45) HCAR2ALDH1A1HAO1GPR84
SCHEMBL7426789 0.66 HCAR2 (0.44) HCAR2KDM4ECYP2C19HSD17B10HAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005011609-A2 TRIAZOLOPURINE-BASED TRICYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME BRISTOL-MYERS SQUIBB COMPANY (US) 2005-02-10 WO disclosed
WO-2004075846-A2 PYRAZOLOPURINE-BASED TRICYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME BRISTOL-MYERS SQUIBB COMPANY (US) 2004-09-10 WO disclosed