SCHEMBL6469940

SCHEMBL6469940

Fc1ccc(Br)c(Oc2cccc(Br)c2)c1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 7/20 0.41
POLB P06746 1/20 0.38
HSP90AA1 P07900 1/20 0.38
MAPT P10636 1/20 0.38
EGFR P00533 3/20 0.37
ABCG2 Q9UNQ0 1/20 0.35
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
ATM Q13315 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDR P35968 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6469872 0.80 POLB (0.45) MAOBPOLBHSP90AA1MAPTEGFR
SCHEMBL30593929 0.74 MAOB (0.44) MAOBEGFRABCG2KDRSLC6A2
SCHEMBL6469983 0.73 CYP1A2 (0.41) MAOBPOLBHSP90AA1MAPTEGFR
SCHEMBL457828 0.73 MAOB (0.54) MAOBMAPTEGFRABCG2KDR
SCHEMBL2461156 0.72 MAPT (0.38) POLBHSP90AA1MAPTEGFRKDR
SCHEMBL3842164 0.71 MAOB (0.52) MAOBMAPTEGFRABCG2SLC6A2
SCHEMBL3899847 0.71 MAOB (0.59) MAOBMAPTEGFRABCG2SLC6A2
SCHEMBL30076271 0.70 EGFR (0.42) MAOBMAPTEGFRABCG2CYP1A2
SCHEMBL3891773 0.70 MAOB (0.47) MAOBEGFRABCG2CYP1A2CYP3A4
SCHEMBL17608807 0.70 MAPT (0.41) MAOBPOLBHSP90AA1MAPTSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005077868-A2 CONGENERIC, CHLORINATED, BROMINATED AND/OR IODISED, FLUORINATED AROMATIC COMPOUNDS COMPRISING TWO BENZOL RINGS IN THEIR BASIC STRUCTURE, METHOD FOR THEIR PRODUCTION AND USE THEREOF CHIRON AS (NO) 2005-08-25 WO claimed
WO-2005077868-A2 CONGENERIC, CHLORINATED, BROMINATED AND/OR IODISED, FLUORINATED AROMATIC COMPOUNDS COMPRISING TWO BENZOL RINGS IN THEIR BASIC STRUCTURE, METHOD FOR THEIR PRODUCTION AND USE THEREOF CHIRON AS (NO) 2005-08-25 WO disclosed