SCHEMBL6470376

SCHEMBL6470376

CC(C(=O)C1CCCCC1)c1ccc2c(c1)nc(N)n2CCC(N)=O

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITK Q08881 16/20 0.65
BACE1 P56817 4/20 0.47
INSR P06213 6/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6469077 0.81 ITK (0.50) ITKBACE1INSR
SCHEMBL6469297 0.79 BACE1 (0.48) ITKBACE1INSR
SCHEMBL5576415 0.79 ITK (0.69) ITKINSR
SCHEMBL6469021 0.79 ITK (0.74) ITKINSR
SCHEMBL6414034 0.74 TLR8 (0.63) ITKBACE1INSR
SCHEMBL6023568 0.73 BACE1 (0.48) ITKBACE1INSR
SCHEMBL6261949 0.72 BACE1 (0.53) ITKBACE1INSR
SCHEMBL6023576 0.71 KMT2A (0.56)
SCHEMBL14708868 0.71 BACE1 (0.52) ITKBACE1
SCHEMBL6023581 0.71 ITK (0.59) ITKBACE1INSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050176792-A1 Ketone substituted benzimidazole compounds BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-08-11 US disclosed
WO-2005070420-A1 1H-BENZIMIDAZOL-2-YL-BENZAMIDE DERIVATIVES AND RELATED COMPOUNDS AS ITK INHIBITORS (INTERLEUKIN-2-INDUCIBLE T CELL KINASE) FOR THE TREATMENT OF INFLAMMATION, IMMUNOLOGICAL AND ALLERGIC DISORDERS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-08-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050176792-A1 Ketone substituted benzimidazole compounds ITK, BLK, BCKDK ITK 1/4885BACE1 1492/4885INSR 518/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.