SCHEMBL6471507

SCHEMBL6471507

Cc1[nH]c(=O)c(Cl)c(OCc2ccc(F)cc2F)c1Cc1ccc(C(=O)NCC(C)(C)O)cc1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 13/20 0.41
MAPK11 Q15759 2/20 0.40
SNCA P37840 1/20 0.38
NAMPT P43490 1/20 0.38
AR P10275 1/20 0.38
MAOB P27338 1/20 0.37
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6533872 0.91 MAPK14 (0.44) MAPK14MAPK11
SCHEMBL4377468 0.86 MAPK14 (0.43) MAPK14MAPK11ARMAOB
SCHEMBL6471580 0.85 MAPK14 (0.45) MAPK14MAOB
SCHEMBL6471516 0.85 MAPK14 (0.51) MAPK14MAOB
SCHEMBL6471919 0.84 MAPK14 (0.40) MAPK14MAOB
SCHEMBL6472203 0.83 MAPK14 (0.57) MAPK14MAOB
SCHEMBL6471631 0.82 MAPK14 (0.59) MAPK14MAPK11
Hydrochloric Acid SCHEMBL6473516 0.81 MAPK14 (0.39) MAPK14MAOB
SCHEMBL6472893 0.80 MAPK14 (0.51) MAPK14MAPK11
Hydrochloric Acid SCHEMBL6470993 0.80 MAPK14 (0.44) MAPK14MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3691620-A1 P38 KINASE INHIBITORS REDUCE DUX4 AND DOWNSTREAM GENE EXPRESSION FOR THE TREATMENT OF FSHD Fulcrum Therapeutics, Inc. (US) 2020-08-12 EP disclosed
WO-2019071147-A1 P38 KINASE INHIBITORS REDUCE DUX4 AND DOWNSTREAM GENE EXPRESSION FOR THE TREATMENT OF FSHD Fulcrum Therapeutics, Inc. (US) 2019-04-11 WO disclosed
WO-2005018557-A2 SUBSTITUTED PYRIDINONES PHARMACIA CORPORATION (US) 2005-03-03 WO disclosed