SCHEMBL6475284

SCHEMBL6475284

COC(=O)c1ccc(-c2ccc(OC(C)CNS(=O)(=O)C(C)C)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 6/20 0.53
SMN1; SMN2 Q16637 1/20 0.48
CA1 P00915 5/20 0.48
CA2 P00918 5/20 0.48
CA12 O43570 4/20 0.48
CA9 Q16790 4/20 0.48
CA14 Q9ULX7 4/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
STS P08842 1/20 0.46
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.43
PLAU P00749 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6480644 0.91 GRIA4 (0.66) GRIA4MEN1KMT2AMTNR1AMTNR1B
SCHEMBL6482318 0.90 GRIA4 (0.53) GRIA4MTNR1AMTNR1BMAPT
SCHEMBL6481796 0.88 GRIA4 (0.50) GRIA4CA1CA2CA12CA9
SCHEMBL6482156 0.87 MTNR1A (0.52) GRIA4MTNR1AMTNR1B
SCHEMBL6475287 0.85 SMN1; SMN2 (0.47) GRIA4SMN1; SMN2CA1CA2CA12
SCHEMBL6475291 0.85 GRIA4 (0.62) GRIA4MTNR1AMTNR1BMAPT
SCHEMBL6474389 0.85 GRIA4 (0.62) GRIA4MEN1KMT2AMTNR1AMTNR1B
SCHEMBL6475304 0.83 GRIA4 (0.47) GRIA4CA1CA2MTNR1AMTNR1B
SCHEMBL6472657 0.83 GRIA4 (0.47) GRIA4CA1CA2MTNR1AMTNR1B
SCHEMBL6482776 0.83 GRIA4 (0.49) GRIA4SMN1; SMN2CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6911476-B2 Sulfonamide derivatives ELI LILLY AND COMPANY (US) 2005-06-28 US claimed
US-20030225266-A1 Sulfonamide derivatives ELI LILLY AND COMPANY 2003-12-04 US claimed
EP-1265857-A1 SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2002-12-18 EP claimed
WO-2001068592-A1 SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2001-09-20 WO claimed
US-6911476-B2 Sulfonamide derivatives ELI LILLY AND COMPANY (US) 2005-06-28 US disclosed
US-20030225266-A1 Sulfonamide derivatives ELI LILLY AND COMPANY 2003-12-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225266-A1 Sulfonamide derivatives GRIN2A, GRM2, GRIA2 GRIA4 6/4885SMN1; SMN2 534/4885CA1 1199/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.