SCHEMBL6476780

SCHEMBL6476780

COc1ccc(-c2ccccc2)c2sc(NC(=O)c3ccc(CN4CCNCC4)cc3)nc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.52
HDAC6 Q9UBN7 1/20 0.52
ADORA2A P29274 5/20 0.48
ADORA2B P29275 5/20 0.48
ADORA1 P30542 5/20 0.48
MAPT P10636 4/20 0.48
IKBKE Q14164 1/20 0.47
TBK1 Q9UHD2 1/20 0.47
DUSP3 P51452 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
TP53 P04637 1/20 0.46
LMNA P02545 2/20 0.46
HPGD P15428 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
USP2 O75604 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CHRM3 P20309 1/20 0.45
CHRM4 P08173 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3048007 0.99 HDAC1 (0.51) HDAC1HDAC6ADORA2AADORA2BADORA1
SCHEMBL3047088 0.97 HDAC1 (0.49) HDAC1HDAC6ADORA2AADORA2BADORA1
Hydrochloric Acid SCHEMBL3054603 0.96 HDAC1 (0.49) HDAC1HDAC6ADORA2AADORA2BADORA1
SCHEMBL5036546 0.92 HDAC1 (0.54) HDAC1HDAC6ADORA2AADORA2BADORA1
Hydrochloric Acid SCHEMBL3048068 0.91 HDAC1 (0.54) HDAC1HDAC6ADORA2AADORA2BADORA1
SCHEMBL6485716 0.91 HDAC1 (0.54) HDAC1HDAC6ADORA2AADORA2BADORA1
SCHEMBL6481675 0.91 ALK (0.54) HDAC1HDAC6ADORA2AADORA2BADORA1
Hydrochloric Acid SCHEMBL3051261 0.91 TRPV4 (0.53) HDAC1HDAC6ADORA2AADORA2BADORA1
SCHEMBL3039082 0.91 HDAC1 (0.53) HDAC1HDAC6ADORA2AADORA2BADORA1
Hydrochloric Acid SCHEMBL3053390 0.90 KIT (0.53) HDAC1HDAC6ADORA2AADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6963000-B2 Benzothiazole derivatives with activity as adenosine receptor ligands HOFFMAN-LA ROCHE INC. (US) 2005-11-08 US claimed