SCHEMBL6476840

SCHEMBL6476840

NC(Cc1ccc(Cl)cc1)C(=O)N1CCC(Cc2cccs2)(C2CCCC2)CC1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MC4R P32245 6/20 0.60
MC3R P41968 1/20 0.60
MC1R Q01726 1/20 0.60
DPP7 Q9UHL4 3/20 0.46
DPP4 P27487 2/20 0.46
FAP Q12884 1/20 0.46
DPP8 Q6V1X1 1/20 0.46
DPP9 Q86TI2 1/20 0.46
AKT1 P31749 9/20 0.43
AKT2 P31751 1/20 0.42
AKT1S1 Q96B36 1/20 0.42
AKT3 Q9Y243 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6199494 0.99 MC4R (0.62) MC4RMC3RMC1RDPP7DPP4
SCHEMBL6477249 0.96 MC4R (0.55) MC4RMC3RMC1RDPP7DPP4
SCHEMBL6476088 0.83 MC4R (0.70) MC4RMC3RMC1RDPP7DPP4
SCHEMBL6476091 0.83 MC4R (0.70) MC4RMC3RMC1RDPP7DPP4
SCHEMBL6483327 0.82 MC4R (0.68) MC4RMC3RMC1RDPP7DPP4
SCHEMBL6949567 0.81 MC4R (0.50) MC4RMC3RMC1RDPP7DPP8
SCHEMBL6197883 0.81 MC4R (0.70) MC4RMC3RMC1RDPP7DPP4
SCHEMBL6476760 0.79 MC4R (0.60) MC4RMC3RMC1RDPP7DPP4
SCHEMBL6476767 0.79 MC4R (0.60) MC4RMC3RMC1RAKT1
SCHEMBL6476771 0.79 MC4R (0.60) MC4RMC3RMC1RAKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050239835-A1 Melanocortin receptor ligands EBETINO FRANK H 2005-10-27 US disclosed
US-20040010010-A1 Melanocortin receptor ligands PROCTER & GAMBLE COMPANY, THE 2004-01-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050239835-A1 Melanocortin receptor ligands MC1R, MC4R, MC3R MC4R 2/4885MC3R 3/4885MC1R 1/4885
US-20040010010-A1 Melanocortin receptor ligands MC1R, MC4R, MC5R MC4R 2/4885MC3R 4/4885MC1R 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.