SCHEMBL6481358

SCHEMBL6481358

CC(C)C[C@H](N)C(=O)N[C@@H](Cc1ccc(OC(=O)N2CCOCC2)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 8/20 0.49
RAB9A P51151 2/20 0.46
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
MMP1 P03956 1/20 0.42
ITGB1 P05556 1/20 0.42
ITGA4 P13612 1/20 0.42
ITGB7 P26010 1/20 0.42
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PSMB8 P28062 1/20 0.41
YAP1 P46937 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6686538 1.00 CACNA1B (0.49) CACNA1BRAB9ACYP1A2CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL7539648 0.99 CACNA1B (0.48) CACNA1BRAB9ACYP1A2CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL6473882 0.99 CACNA1B (0.48) CACNA1BRAB9ACYP1A2CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL6691605 0.90 CACNA1B (0.45) CACNA1BKMT2AMEN1MMP1ITGB1
Hydrochloric Acid SCHEMBL6691609 0.90 CACNA1B (0.45) CACNA1BKMT2AMEN1MMP1ITGB1
SCHEMBL7536860 0.87 CACNA1B (0.50) CACNA1BKMT2AMEN1MMP1ITGB1
SCHEMBL6479164 0.87 CACNA1B (0.50) CACNA1BKMT2AMEN1MMP1ITGB1
Hydrochloric Acid SCHEMBL6480368 0.86 CACNA1B (0.49) CACNA1BKMT2AMEN1MMP1ITGB1
Hydrochloric Acid SCHEMBL7540812 0.86 CACNA1B (0.49) CACNA1BKMT2AMEN1MMP1ITGB1
SCHEMBL6473757 0.86 CACNA1B (0.46) CACNA1BRAB9ACYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6867192-B1 Compounds useful in the treatment of inflammatory diseases GLAXO GROUP LIMITED (GB) 2005-03-15 US disclosed
EP-1140837-B1 COMPOUNDS USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASES GLAXO GROUP LTD (GB) 2004-08-18 EP disclosed
EP-1140837-A1 COMPOUNDS USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2001-10-10 EP disclosed
WO-2000037444-A1 COMPOUNDS USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2000-06-29 WO disclosed