SCHEMBL6481483

SCHEMBL6481483

CC1(C)OB(c2ccc(OC(=O)O)c(F)c2)OC1(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.46
LIPG Q9Y5X9 5/20 0.43
LPL P06858 4/20 0.43
F2 P00734 2/20 0.41
F11 P03951 2/20 0.41
PRSS1 P07477 2/20 0.41
PRSS2 P07478 2/20 0.41
PRSS3 P35030 2/20 0.41
P4HB P07237 1/20 0.39
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA9 Q16790 3/20 0.38
BACE1 P56817 1/20 0.38
BACE2 Q9Y5Z0 1/20 0.38
AAK1 Q2M2I8 1/20 0.38
HIF1A Q16665 3/20 0.37
CSF1R P07333 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28929431 0.87 ROCK1 (0.45) ROCK1LIPGLPLF2F11
SCHEMBL6183441 0.84 ROCK1 (0.45) ROCK1LIPGLPLF2F11
SCHEMBL25177249 0.82 AAK1 (0.45) ROCK1LIPGLPLF2F11
SCHEMBL31264705 0.81 ROCK1 (0.47) ROCK1LIPGLPLBACE1BACE2
SCHEMBL31264645 0.81 ROCK1 (0.47) ROCK1LIPGLPLBACE1BACE2
SCHEMBL1643648 0.81 HIF1A (0.41) LIPGLPLF2F11PRSS1
SCHEMBL142144 0.80 LPL (0.49) ROCK1LIPGLPLCA1CA2
SCHEMBL31264766 0.80 ROCK1 (0.47) ROCK1LMNAMAPK1HTTRAB9A
SCHEMBL1130871 0.78 ROCK1 (0.48) ROCK1LIPGLPLF2F11
SCHEMBL4366318 0.77 LPL (0.47) ROCK1LIPGLPLP4HBCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6919343-B2 N-biphenyl(substituted methyl) aminocycloalkane-carboxamide derivatives MERCK & CO., INC. (US) 2005-07-19 US disclosed