SCHEMBL648259

SCHEMBL648259

CCOc1cccc(CN(Cc2ccc3c(c2)OCCO3)Cc2c(Cl)nc(-c3ccccc3)n2CCN2CCCCC2)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
MAPK1 P28482 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
C5AR1 P21730 1/20 0.39
F2R P25116 8/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TSHR P16473 1/20 0.36
ESR1 P03372 1/20 0.36
CYP2D6 P10635 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
GAA P10253 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL650618 0.95 ALDH1A1 (0.41) ALDH1A1MAPK1OPRM1OPRD1C5AR1
SCHEMBL649494 0.91 C5AR1 (0.44) ALDH1A1MAPK1OPRM1OPRD1C5AR1
SCHEMBL648633 0.89 C5AR1 (0.50) ALDH1A1MAPK1OPRM1OPRD1C5AR1
SCHEMBL650106 0.87 C5AR1 (0.40) ALDH1A1MAPK1OPRM1OPRD1C5AR1
SCHEMBL650054 0.86 C5AR1 (0.49) C5AR1TSHRGAAKDM4E
SCHEMBL1913026 0.85 C5AR1 (0.56) C5AR1TSHR
SCHEMBL648110 0.84 C5AR1 (0.49) ALDH1A1MAPK1OPRM1OPRD1C5AR1
SCHEMBL649431 0.84 C5AR1 (0.44) ALDH1A1MAPK1OPRM1OPRD1C5AR1
SCHEMBL650039 0.83 C5AR1 (0.49) ALDH1A1MAPK1OPRM1OPRD1C5AR1
SCHEMBL1913083 0.83 C5AR1 (0.43) ALDH1A1MAPK1OPRM1OPRD1C5AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119665-B2 Aryl imidazoles and related compounds as C5a receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-02-21 US disclosed
US-7186734-B2 Aryl imidazoles and related compounds as C5a receptor modulators NEUROGEN CORPORATION (US) 2007-03-06 US disclosed
US-7186734-B2 Aryl imidazoles and related compounds as C5a receptor modulators NEUROGEN CORPORATION (US) 2007-03-06 US disclosed
US-7186734-B2 Aryl imidazoles and related compounds as C5a receptor modulators NEUROGEN CORPORATION (US) 2007-03-06 US disclosed