SCHEMBL6484128

SCHEMBL6484128

COc1ccc(-c2ccccc2)c2sc(NC(=O)c3ccc(CNCc4cccs4)cc3)nc12

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.51
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
CHRM4 P08173 3/20 0.47
DUSP3 P51452 2/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C19 P33261 1/20 0.46
ADORA2A P29274 8/20 0.46
ADORA2B P29275 8/20 0.46
ADORA1 P30542 8/20 0.46
NPSR1 Q6W5P4 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3049704 0.99 HDAC1 (0.50) HDAC1HDAC8HDAC6CHRM4DUSP3
SCHEMBL6476277 0.91 DUSP3 (0.53) CHRM4DUSP3ADORA2AADORA2BADORA1
Hydrochloric Acid SCHEMBL3045899 0.90 DUSP3 (0.53) CHRM4DUSP3ADORA2AADORA2BADORA1
SCHEMBL3047875 0.90 CHRM4 (0.57) CHRM4DUSP3ADORA2AADORA2BADORA1
Hydrochloric Acid SCHEMBL3050847 0.89 CHRM4 (0.56) CHRM4DUSP3ADORA2AADORA2BADORA1
SCHEMBL6477408 0.88 DUSP3 (0.52) CHRM4DUSP3ADORA2AADORA2BADORA1
SCHEMBL3055622 0.87 DUSP3 (0.51) CHRM4DUSP3ADORA2AADORA2BADORA1
Hydrochloric Acid SCHEMBL3050899 0.87 DUSP3 (0.51) CHRM4DUSP3ADORA2AADORA2BADORA1
Hydrochloric Acid SCHEMBL3058132 0.86 DUSP3 (0.50) CHRM4DUSP3ADORA2AADORA2BADORA1
SCHEMBL3057471 0.86 DUSP3 (0.50) CHRM4DUSP3MAPTADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6963000-B2 Benzothiazole derivatives with activity as adenosine receptor ligands HOFFMAN-LA ROCHE INC. (US) 2005-11-08 US claimed