SCHEMBL6484767

SCHEMBL6484767

CCCNCc1ccc(C(=O)Nc2nc3c(OC)ccc(-c4ccccc4)c3s2)cc1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DUSP3 P51452 2/20 0.50
ADORA2A P29274 11/20 0.48
ADORA2B P29275 11/20 0.48
ADORA1 P30542 11/20 0.48
CHRM4 P08173 2/20 0.48
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3039089 0.99 DUSP3 (0.49) DUSP3ADORA2AADORA2BADORA1CHRM4
SCHEMBL3055622 0.94 DUSP3 (0.51) DUSP3ADORA2AADORA2BADORA1CHRM4
Hydrochloric Acid SCHEMBL3058132 0.93 DUSP3 (0.50) DUSP3ADORA2AADORA2BADORA1CHRM4
SCHEMBL3057471 0.93 DUSP3 (0.50) DUSP3ADORA2AADORA2BADORA1CHRM4
SCHEMBL6477408 0.93 DUSP3 (0.52) DUSP3ADORA2AADORA2BADORA1CHRM4
SCHEMBL6476277 0.93 DUSP3 (0.53) DUSP3ADORA2AADORA2BADORA1CHRM4
Hydrochloric Acid SCHEMBL3044579 0.92 DUSP3 (0.49) DUSP3ADORA2AADORA2BADORA1CHRM4
Hydrochloric Acid SCHEMBL3050899 0.92 DUSP3 (0.51) DUSP3ADORA2AADORA2BADORA1CHRM4
Hydrochloric Acid SCHEMBL3045899 0.92 DUSP3 (0.53) DUSP3ADORA2AADORA2BADORA1CHRM4
SCHEMBL6485433 0.90 HDAC1 (0.50) DUSP3ADORA2AADORA2BADORA1CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6963000-B2 Benzothiazole derivatives with activity as adenosine receptor ligands HOFFMAN-LA ROCHE INC. (US) 2005-11-08 US claimed