SCHEMBL6485940

SCHEMBL6485940

CCOC(=O)CN(CC(F)(F)F)c1ccc(C(O)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.59
AR P10275 1/20 0.53
NR1H3 Q13133 7/20 0.52
NR1H2 P55055 6/20 0.52
MLYCD O95822 8/20 0.47
RORC P51449 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
GAA P10253 1/20 0.46
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6484353 0.90 LMNA (0.61) LMNANR1H3NR1H2MLYCDSMN1; SMN2
SCHEMBL6486759 0.84 LMNA (0.55) LMNANR1H3NR1H2MLYCDRORC
SCHEMBL6488084 0.83 NR1H2 (0.67) LMNANR1H3NR1H2MLYCDRORC
SCHEMBL6486223 0.83 NR1H2 (0.54) LMNANR1H3NR1H2MLYCDRORC
SCHEMBL6501262 0.83 NR1H2 (0.55) LMNANR1H3NR1H2MLYCD
SCHEMBL6485130 0.83 LMNA (0.67) LMNANR1H3NR1H2MLYCDSMN1; SMN2
SCHEMBL6486856 0.81 NR1H2 (0.52) LMNANR1H3NR1H2MLYCD
SCHEMBL6496268 0.81 NR1H2 (0.63) LMNANR1H3NR1H2MLYCDRORC
SCHEMBL6211393 0.81 NR1H2 (0.53) LMNANR1H3NR1H2MLYCDRORC
SCHEMBL6486621 0.80 NR1H2 (0.51) LMNANR1H3NR1H2MLYCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6900244-B2 Anilino liver X-receptor modulators PHARMACIA CORPORATION (US) 2005-05-31 US claimed
US-20040087632-A1 Controlling metabolism of lipids, cholesterol PHARMACIA CORPORATION 2004-05-06 US claimed
US-6900244-B2 Anilino liver X-receptor modulators PHARMACIA CORPORATION (US) 2005-05-31 US disclosed
US-20040087632-A1 Controlling metabolism of lipids, cholesterol PHARMACIA CORPORATION 2004-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040087632-A1 Controlling metabolism of lipids, cholesterol NR1H2, NR1H3, SREBF1 LMNA 2466/4885AR 586/4885NR1H3 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.